NEW LIGANDS OF CANNACBINOID RECEPTORS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND METHOD FOR PRODUCING THEREOF Russian patent published in 2011 - IPC C07D231/54 C07D401/12 C07D405/12 C07D409/12 A61K31/416 A61P25/00 

Abstract RU 2420518 C2

FIELD: medicine.

SUBSTANCE: present invention presents new compounds which are modulators of cannabinoid receptors, particularly modulators of cannabinoid receptors 1 (CB1) or cannabinoid receptors 2 (CB2), and an application thereof for treating diseases, conditions and/or disorders regulated by a cannabinoid receptor (such as painful sensations, neurodegenerative disorders, ingestion disorders, weight loss or weight control and obesity), as well as based pharmaceutical compositions. New compounds are characterised by graphic formulas

in which radicals and groups have the values specified in the patent claim.

EFFECT: higher efficiency of applying the composition.

55 cl, 13 tbl, 3 dwg, 802 ex

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Authors

Matappala-Niappan Meijappan

Balasubramanian Gopalan

Gallapalli Srinivas

Dzhoshi Neelima Khajratkar

Narajanan Shridkhar

Dates

2011-06-10Published

2006-06-01Filed