QUINAZOLINE DERIVATIVES Russian patent published in 2011 - IPC C07D239/84 A61K31/517 A61P17/00 A61P17/04 A61P37/08 

Abstract RU 2431632 C2

FIELD: chemistry.

SUBSTANCE: disclosed compounds can be used as an antipruritic agent in case of atopic disease such as atopic dermatitis when a steroid medicinal agent is ineffective. In formula R is C1-6 alkoxy, optionally substituted methyoxy, or an amine which is monosubstituted with C1-6 alkyl, where the R-C(=O)- group is bonded in the meta or para-position.

EFFECT: high efficiency of using said compounds.

21 cl, 16 dwg, 4 tbl, 30 ex

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RU 2 431 632 C2

Authors

Mijazaki Kazuki

Kusano Kazutomi

Takase Jasutaka

Asano Osamu

Sirato Manabu

Vakita Khisasi

Isii Naoto

Saeki Takao

Dates

2011-10-20Published

2007-02-20Filed