AZABICYCLO{3,1,0}HEXANE DERIVATIVES USED AS DOPAMINE RECEPTOR D3 MODULATORS Russian patent published in 2011 - IPC C07D403/12 C07D403/14 C07D405/14 C07D409/14 C07D413/14 C07D417/14 A61K31/403 A61P25/00 

Abstract RU 2434011 C2

FIELD: chemistry.

SUBSTANCE: described are novel derivatives of azabicyclo{3,1,0}hexane of general formula (I) or pharmaceutically acceptable salts thereof (values of radicals are given in the claim), synthesis method thereof, intermediate compounds, a pharmaceutical composition and use of the novel compounds in therapy as dopamine receptor D3 modulators, for example, for treating drug dependence or as antipsychotic agents.

EFFECT: improved properties of the derivatives.

34 cl, 122 ex

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RU 2 434 011 C2

Authors

Arista Luka

Bonanomi Dzhordzho

Kapelli Anna Marija

Damiani Federika

Di Fabio Romano

Dzhentile Gabriella

Khamprekht Diter Vol'Fgang

Mikeli Fabritsio

Tarsi Luka

Tedesko Dzhovanna

Terreni Sil'Vija

Dates

2011-11-20Published

2005-02-21Filed