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(19)

(11)

2 440 992

(13)

(51)

IPC

C07D241/24(2006-01-01)

C07D401/12(2006-01-01)

C07D403/12(2006-01-01)

A61K31/4439(2006-01-01)

A61K31/497(2006-01-01)

A61P3/00(2006-01-01)

A61P3/04(2006-01-01)

A61P3/10(2006-01-01)

(21) (22)

Application

2009114802/04, 2007-10-25

(24)

Start date

2007-10-25

(22)

Actual filing date

2007-10-25

(45)

Published

2012-01-27

(72)

Inventor

Martin Nataniehl' DzhordzhMakkerrecher DarrenPajk Kurt GordonUoring Majkl Dzhejms

(73)

Holder

Astrazeneka Ab

BENZOYLAMINOHETEROCYCLYL COUMPOUNDS AS GLUCOKINASE (GLK) ACTIVATORS Russian patent published in 2012 - IPC C07D241/24 C07D401/12 C07D403/12 A61K31/4439 A61K31/497 A61P3/00 A61P3/04 A61P3/10

Abstract RU 2440992 C2

FIELD: chemistry.

SUBSTANCE: present invention refers to the compound 5-[3-[(2S)-1-(difluoromethoxy)-propane-2-yl]-oxy-5-[(5-methylpyrazin-2-yl)-carbamoyl]]phenoxy]-N,N-dimethyl-pyrazine-2-carboxamide. The invention also refers to a pharmaceutical composition, and also to application of the compound under cl.1.

EFFECT: making the new biologically active compounds showing GLK (glucokinase) activator activity.

5 cl, 6 ex, 2 tbl, 2 dwg

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RU 2 440 992 C2

Authors

Martin Nataniehl' Dzhordzh

Makkerrecher Darren

Pajk Kurt Gordon

Uoring Majkl Dzhejms

Dates

2012-01-27—Published

2007-10-25—Filed