SERINE PROTEASE INHIBITORS Russian patent published in 2012 - IPC C07K5/10 A61K38/07 A61P31/14 

Abstract RU 2441020 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a mixture of diastereomeric compounds where C* denotes a mixture of R- and S-isomers; and the R-isomer constitutes over 50% of the mixture with respect to the S-isomer in the C* position.

EFFECT: obtained mixture is effective for inhibiting serine protease.

16 cl, 8 tbl, 6 dwg, 9 ex

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RU 2 441 020 C2

Authors

Lajonz Stiv

Perni Robert B.

Dates

2012-01-27Published

2006-08-01Filed