AZETINE COMPOUNDS AS OREXIN RECEPTOR ANTAGONISTS Russian patent published in 2012 - IPC C07D405/12 C07D417/14 C07D515/04 A61K31/397 A61P25/00 

Abstract RU 2447070 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: present invention refers to a compound of formula

wherein R1, R2 and X are those as specified in cl.1 of the patent claim, or its pharmaceutically acceptable salt, as well as using such compound or its pharmaceutically acceptable salt for preparing a drug preparation for prevention and treatment of all types of sleeping, eating or drinking disorders.

EFFECT: preparing the new azetidine compounds showing activity of orexin receptor antagonists.

12 cl, 112 ex, 1 tbl

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RU 2 447 070 C2

Authors

Ehssaui Amed

Boss Kristof

Gude Markus

Kobershtajn Ral'F

Zifferlen T'Erri

Dates

2012-04-10Published

2007-08-15Filed