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2 449 996

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(51)

IPC

C07D261/02(2006-01-01)

C07D413/12(2006-01-01)

C07D413/14(2006-01-01)

A61K31/42(2006-01-01)

A61K31/422(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2009121808/04, 2007-11-14

(24)

Start date

2007-11-14

(22)

Actual filing date

2007-11-14

(45)

Published

2012-05-10

(72)

Inventor

Kastro Al'Fredo S.Kholson Ehduard B.Khopkins Brajan T.Kouni Naj O.Snajder Daniel A.Tibbitts Tomas T.

(73)

Holder

Infiniti Diskaveri, Ink.

COMPOUNDS AND METHODS FOR INHIBITING Bcl PROTEIN INTERACTION WITH BINDING PARTNERS Russian patent published in 2012 - IPC C07D261/02 C07D413/12 C07D413/14 A61K31/42 A61K31/422 A61P35/00

Abstract RU 2449996 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to compounds specified in cl. 1, and also to a pharmaceutical composition possessing binding activity with respect to Bcl proteins, to applying the declared compounds for preparing a drug for treating cancer and for treating a bcl-mediated disorder.

EFFECT: use of the compounds as Bcl protein inhibitors.

18 cl, 2 tbl, 41 ex

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RU 2 449 996 C2

Authors

Kastro Al'Fredo S.

Kholson Ehduard B.

Khopkins Brajan T.

Kouni Naj O.

Snajder Daniel A.

Tibbitts Tomas T.

Dates

2012-05-10—Published

2007-11-14—Filed