SOLUBLE C5aR ANTAGONISTS Russian patent published in 2021 - IPC C07D211/60 C07D401/10 A61K31/451 

Abstract RU 2748260 C2

FIELD: biochemistry.

SUBSTANCE: invention relates to compounds of Formula (I):

in which R1 is selected from a group consisting of H,

R2 is selected from a group consisting of H,

R3 is H, or ; wherein two of R1, R2 and R3 are H, and one of R1, R2 and R3 differs from H, or its pharmacologically acceptable salts modulating C5a receptor. Pharmaceutical compositions containing such compounds and treatment methods are also described.

EFFECT: compounds and pharmaceutical compositions containing such compounds can be used in medicine.

25 cl, 2 dwg, 25 ex

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RU 2 748 260 C2

Authors

Fan, Pinchen

Krasinski, Entoni

Mali, Venkat, Reddi

Myao, Shichan

Punna, Srinivas

Sun, Yan

Stella, Valentino, Dzh.

Tszen, Ibin

Chzhan, Penli

Dates

2021-05-21Published

2017-04-03Filed