4-(1-AMINOETHYL)CYCLOHEXYLAMINE DERIVATIVES Russian patent published in 2012 - IPC C07D215/14 C07D471/04 A61K31/4375 A61P31/04 

FIELD: chemistry.

SUBSTANCE: invention relates to novel 4-(1-aminoethyl)cyclohexylamine derivatives of general formula or pharmaceutically acceptable salts of such a compound, wherein R⁰ represents H or OH; R¹ represents an alkoxy group; U and W represent N, V represents CH and R² represents H or F, or U and V represent CH, W represents N and R² represents H or F, or U and V represent N, W represents CH and R² represents H, or U represents N, V represents CH, W represents CR^a and R² represents H; R^a represents CH₂OH or alkoxycarbonyl; A represents the group CH=CH-B or a binuclear heterocyclic system D; B represents a mono- or di-substituted phenyl group wherein the substitutes are halogen atoms; D represents either a group , wherein Z represents CH or N, and Q represents O or S, or a group . The invention also relates to a pharmaceutical composition based on the compound of formula (I) and to use of the compound of formula (I).

EFFECT: novel derivatives having antibacterial activity are obtained.

12 cl, 21 ex