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(19)

RU

(11)

2 465 275

(13)

C2

(51)

IPC

C07D471/04(2006-01-01)

C07D487/04(2006-01-01)

A61K31/4375(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2009128186/04, 2007-12-21

(24)

Start date

2007-12-21

(22)

Actual filing date

2007-12-21

(45)

Published

2012-10-27

(72)

Inventor

Berdini ValerioBezong Gilbert EhbajKallagan OuehnKarr Marija GratsijaKongriv Majlz StjuartDzhill Ehdrian LiehmGriffits-Dzhounz Sharlott MehriMehdin EhndrjuMjurrej Kristofer Uill'JamNidzhar Radzhdip KaurO'Brajen Majkl AlistehrPajk EhndrjuSaksti GordonTehjlor Richard DehvidVikerstaff Ehmma

(73)

Holder

Asteks Terap'Jutiks Limited

BICYCLIC AMINE DERIVATIVES AS TYROSINE KINASE INHIBITORS Russian patent published in 2012 - IPC C07D471/04 C07D487/04 A61K31/4375 A61P35/00 

Abstract RU 2465275 C2

FIELD: chemistry.

SUBSTANCE: invention relates to novel bicyclic heterocyclic derivatives, which are compounds of formula where values of X1-X5, A, B, R1, R2, q are given in claim 1, as well as pharmaceutical compositions containing said compounds, and use of said compounds to treat cancer.

EFFECT: high efficiency of treatment.

22 cl, 43 ex

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RU 2 465 275 C2

Authors

Berdini Valerio

Bezong Gilbert Ehbaj

Kallagan Ouehn

Karr Marija Gratsija

Kongriv Majlz Stjuart

Dzhill Ehdrian Liehm

Griffits-Dzhounz Sharlott Mehri

Mehdin Ehndrju

Mjurrej Kristofer Uill'Jam

Nidzhar Radzhdip Kaur

O'Brajen Majkl Alistehr

Pajk Ehndrju

Saksti Gordon

Tehjlor Richard Dehvid

Vikerstaff Ehmma

Dates

2012-10-27—Published

2007-12-21—Filed

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