Patenton — panteon of patents

(19)

RU

(11)

2 465 275

(13)

C2

(51)

IPC

C07D471/04(2006-01-01)

C07D487/04(2006-01-01)

A61K31/4375(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2009128186/04, 2007-12-21

(24)

Start date

2007-12-21

(22)

Actual filing date

2007-12-21

(45)

Published

2012-10-27

(72)

Inventor

Berdini ValerioBezong Gilbert EhbajKallagan OuehnKarr Marija GratsijaKongriv Majlz StjuartDzhill Ehdrian LiehmGriffits-Dzhounz Sharlott MehriMehdin EhndrjuMjurrej Kristofer Uill'JamNidzhar Radzhdip KaurO'Brajen Majkl AlistehrPajk EhndrjuSaksti GordonTehjlor Richard DehvidVikerstaff Ehmma

(73)

Holder

Asteks Terap'Jutiks Limited

BICYCLIC AMINE DERIVATIVES AS TYROSINE KINASE INHIBITORS Russian patent published in 2012 - IPC C07D471/04 C07D487/04 A61K31/4375 A61P35/00 

Abstract RU 2465275 C2

FIELD: chemistry.

SUBSTANCE: invention relates to novel bicyclic heterocyclic derivatives, which are compounds of formula where values of X1-X5, A, B, R1, R2, q are given in claim 1, as well as pharmaceutical compositions containing said compounds, and use of said compounds to treat cancer.

EFFECT: high efficiency of treatment.

22 cl, 43 ex

Similar patents RU2465275C2

Title Year Author Number
IMIDAZOPYRIDINE DERIVATIVES AS INHIBITORS OF RECEPTOR TYROSINE KINASES 2009
  • Uill'Jams Brajan Dzhon
  • Berdini Valerio
  • Karr Marija Gratsija
  • Kongriv Majlz Stjuart
  • Frederikson Martin
  • Griffits-Dzhounz Sharlott Mehri
  • Khamlett Kristofer Charl'Z Frederik
  • Mehdin Ehndrju
  • Mjurrej Kristofer Uill'Jam
  • Benning Radzhip Kaur
  • Saksti Gordon
  • Vikerstaff Ehmma
  • Vudkhehd Ehndrju Dzhejms
  • Vudkhehd Stiven Dzhon
  • Frejn Ehddi Zhan Ehdgar
  • Govarts Tom Kornelis Khortense
  • Anzhibo Patrik Rene
 RU2518089C2
BICYCLIC HETEROCYCLIC COMPOUNDS AS FGFR INHIBITORS 2007
  • Berdini Valerio
  • Bezong Gilbert Ehbaj
  • Kallagan Ouehn
  • Karr Marija Gratsija
  • Kongriv Majlz Stjuart
  • Dzhill Ehdrian Liehm
  • Griffits-Dzhounz Sharlott Mehri
  • Mehdin Ehndrju
  • Mjurrej Kristofer Uill'Jam
  • Nidzhar Radzhdip Kaur
  • O'Brajen Majkl Alistehr
  • Pajk Ehndrju
  • Saksti Gordon
  • Tehjlor Richard Dehvid
  • Vikerstaff Ehmma
 RU2466130C2
POLYCYCLIC AGENTS FOR TREATING RESPIRATORY SYNCYTIAL VIRAL INFECTIONS 2004
  • Bond Sajlas
  • Sanford Vanessa Ann
  • Lambert Dzhon Nikolas
  • Lim Chin Ju.
  • Mitchell Dzheffri Piter
  • Drehffan Ehlister Dzhordzh
  • Nirn Roland Genri
 RU2422444C2
PIPERIDINE DERIVATIVES 2011
  • Baumann Karlkhajnts
  • Flor Aleksandr
  • Getshi Ehrvin
  • Grin Ljuk
  • Zholidon Siniz
  • Knust Khenner
  • Limberg An'Ja
  • Luehbbers Tomas
  • Tomas Ehndrju
 RU2554353C2
PYRASOLE[3,4-b]PYRIDINE COMPOUNDS AND THEIR APPLICATION AS PHOSPHODIESTERASE INHIBITORS 2003
  • Allen Dejvid Dzhordzh
  • Kou Dajan Mehri
  • Kuk Karolin Mehri
  • Kuper Ehntoni Uil'Jam Dzhejms
  • Doul Majkl Dehnnis
  • Ehdlin Kristofer Dejvid
  • Khehmblin Dzhuli Nikol'
  • Dzhonson Martin Redpat
  • Dzhounz Pol Spenser
  • Lindvall Mika Kristian
  • Mitchell Sharlotta Dzhejn
  • Rehdgrehjv Ehlison Dzhudit
 RU2348633C2
AMINOTRIAZOLOPYRIDINES AND USING THEM AS KINASE INHIBITORS 2009
  • Bamaniar Sogole
  • Behjts R. Dzh.
  • Blis Kejt
  • Kalabreze Ehndrju Ehntoni
  • Dehniel Tomas Oran
  • Del'Gado Mersedes
  • Ehl'Sner Jan
  • Ehrdman Pol
  • Far Brjus
  • Fergjuson Gregori
  • Li Brehnden
  • Nadol'Ny Liza
  • Pakard Garrik
  • Papa Patrik
  • Plantevin-Krenitski Veronik
  • Riggs Dzhennifer
  • Roan Patrisija
  • Sankar Sabita
  • Sapienza Dzhon
  • Satokh Esitaka
  • Sloan Viktor
  • Stivens Rehndall
  • Terani Lida
  • Tike Dzhehjehshri
  • Torres Ehduardo
  • Uollehjs Ehndrju
  • Vajtfild Brehndon Uehjd
  • Chzhao Tszintszin
 RU2552642C2
NOVEL COMPOUNDS 2016
  • Kemp Mark Ien
  • Stokli Martin Li
  • Medin Endryu
 RU2734256C2
FLUORINATED LIGANDS FOR TARGETING PERIPHERAL BENZODIAZEPINE RECEPTORS 2007
  • Katsifis Ehndrju
  • Fuks Kristofer Dzhon Redzhinal'D
  • Fam Tien Kuok
  • Gregurik Ivan Damir
  • Mattner Marija Filomena Perejra Soares
 RU2468014C2
PYRIDINES SUBSTITUTED WITH HETEROARYL AND APPLICATION METHODS 2017
  • Altenbakh Robert Dzh.
  • Bogdan Endryu
  • Koti Dyuvanni Petru Diunizu
  • Kauert Marlon D.
  • Gresler Stefen N
  • Kelgtermans Khans
  • Kim Filip R.
  • Van Der Plas Stiven Emil
  • Van Syuetsin
 RU2756743C2
COMPOUNDS BASED ON PYRAZOLOPYRIDINONE 2018
  • Go, Khajbin
  • Van, Chzhao-Kuj
  • Tsin, Lokhen
  • Lyu, Tsyan
  • Cheun, Ving Shun
 RU2806751C2

RU 2 465 275 C2

Authors

Berdini Valerio

Bezong Gilbert Ehbaj

Kallagan Ouehn

Karr Marija Gratsija

Kongriv Majlz Stjuart

Dzhill Ehdrian Liehm

Griffits-Dzhounz Sharlott Mehri

Mehdin Ehndrju

Mjurrej Kristofer Uill'Jam

Nidzhar Radzhdip Kaur

O'Brajen Majkl Alistehr

Pajk Ehndrju

Saksti Gordon

Tehjlor Richard Dehvid

Vikerstaff Ehmma

Dates

2012-10-27—Published

2007-12-21—Filed

download Download PDF read Similar patents