1,3,5-TRISUBSTITUTED TRIAZOLE DERIVATIVE Russian patent published in 2013 - IPC C07D405/14 A61K31/4427 A61P25/10 A61P29/00 

Abstract RU 2476433 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to a new compound of 2-[3-(2,2-difluorobenzo[1,3]dioxol-5-ylamino)-5-(2,6-dimethylpyridin-4-yl)-[1,2,4]triazol4-yl]-N-ethylacetamide and/or pharmaceutically acceptable salts, or hydrate, or solvates, as well as to a method for preparing it; a pharmaceutical composition based on this compound and using its in therapy for prevention and treatment of mental disorders, intellectual disorders or diseases, inflammatory diseases or conditions wherein α7 nicotinic receptor modulation is considered to be favourable. The invention also refers to a product containing such compound and α7-nicotinic receptor agonist.

EFFECT: preparing the compounds applicable in therapy for prevention or treatment of mental disorders, intellectual disorders or diseases, inflammatory diseases or conditions wherein α7 nicotinic receptor modulation is considered to be favourable.

6 cl, 1 tbl, 4 ex

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RU 2 476 433 C2

Authors

Tjuring Jokhannes Vil'Khel'Mus Jokhn F.

Dinklo Teodorus

Lezazh Ann Simon Zhozefin

Dates

2013-02-27Published

2008-10-15Filed