DIPEPTIDE PRODRUGS AND USE THEREOF Russian patent published in 2013 - IPC C07D417/12 C07D417/14 C07D213/85 C07K5/06 A61K31/4418 A61K31/4427 A61K38/05 A61P9/00 

Abstract RU 2486183 C9

FIELD: medicine, pharmaceutics.

SUBSTANCE: application describes prodrugs being 2-amino-6-({[2-(4-chlorophenyl)-1,3-thiazol-4-yl]methyl}thio)-4-[4-(2-hydroxyethoxy)-phenyl]pyridine-3,5-dicarbonitryl derivatives, and a method for preparing them.

EFFECT: invention can find application in treating and/or preventing cardiovascular diseases.

8 cl, 4 tbl, 18 ex

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RU 2 486 183 C9

Authors

Lerkhen Khans-Georg

Krents Ursula

Kel'Denikh Jorg

Didrikhs Nikol'

Kran Tomas

Khirt-Ditrikh Klaudia

Al'Brekht-Kjupper Barbara

Dates

2013-06-27Published

2008-07-23Filed