SUBSTITUTED OXOPYRIDINE DERIVATIVE Russian patent published in 2023 - IPC C07D471/04 A61K31/4427 A61P7/02 

Abstract RU 2792645 C2

FIELD: medicine.

SUBSTANCE: invention relates to 5-({6-amino-2-[4-(5-chlor-2-cyanophenyl)-5-methoxy-2-oxopyridine-1(2H)-yl]-3-methylhexanoyl}amino)pyrazolo[1,5-a]pyridine-3-carboxamide of the formula (I) or to one of its salts.

EFFECT: new compound is obtained, which can be used in medicine as an inhibitor of destructive activity of plasma kallikrein to produce drugs for the treatment and/or prevention of diseases, in particular cardiovascular diseases, preferably thrombotic or thromboembolic disorders and edema, as well as ophthalmic disorders.

3 cl, 3 ex

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RU 2 792 645 C2

Authors

Lobell, Mario

Schirok, Hartmut

Tersteegen, Adrian

Dates

2023-03-22Published

2019-04-03Filed