USE OF 2,4-DIAMINOPYRIMIDINES FOR TREATING ATHEROSCLEROSIS Russian patent published in 2013 - IPC A61K31/5383 A61K31/662 A61P9/10 

Abstract RU 2490015 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to medicine, particularly to pharmaceutical treatment of atherosclerosis and an associated risk of cardiovascular diseases. That is ensured by using the effective amount of a Syk-kinase inhibitor representing N4-(2,2-dimethyl-4-[(dihydrophosphonoxy)methyl]-3-oxo-5-pyrido[1,4]oxazin-6-yl)-5-fluor-K2-(3,4,5-trimethoxyphenyl)-2,4-diamonopyrimidines and a salt thereof.

EFFECT: method provides the substantial size reduction of the atherosclerotic involvements, particularly of the aortic root and arch.

5 ex, 2 tbl, 2 dwg

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RU 2 490 015 C2

Authors

Masuda Ehsteban

Shmitts Jokhen

Dates

2013-08-20Published

2009-02-20Filed