METHOD OF PRODUCING THIOPHENE DERIVATIVE AND INTERMEDIATE PRODUCT THEREOF Russian patent published in 2013 - IPC C07D333/32 C07C319/18 C07C323/56 

Abstract RU 2495877 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a method of producing a thiophene derivative or intermediate product thereof, which can be used as an intermediate product for producing medical and agricultural preparations , where R1 is a C6-10-aryl group (the C6-10 aryl group is unsubstituted or substituted with one or two halogen atoms, one or two C1-10-alkyl groups or C1-10-alkoxy group (the C1-10-alkyl group and C1-10-alkoxy group are unsubstituted or substituted with one or more halogen atoms)), R4 is a C1-3-alkyl group (the C1-3-alkyl group is unsubstituted or substituted with a halogen atom), and X is a leaving group; R2 and R3 are independently a hydrogen atom, C1-6-alkyl group (the C1-6-alky group is unsubstituted or substituted with a halogen atom).

EFFECT: high efficiency of the method.

22 cl, 5 tbl, 58 ex

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RU 2 495 877 C2

Authors

Janagikhara Kazufumi

Umezava Singo

Mijadzi Katsuaki

Dates

2013-10-20Published

2009-02-27Filed