5-HYDROXYMETHYLOXAZOLIN-2-ONE DERIVATIVES FOR TREATING BACTERIAL INTESTINAL DISEASES Russian patent published in 2014 - IPC A61K31/4375 A61P31/04 

Abstract RU 2527769 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to compounds of formula

wherein A means N or CH; and n is equal to 0 or 1; or their pharmaceutically acceptable salts for preventing or treating intestinal diseases caused by a bacterium specified in Clostridium difficile, Clostridium perfringens or Staphylococcus aureus.

EFFECT: present invention possesses a high activity on the agents of intestinal infections, reduces a toxin load, spore production inducing thereby the minimum effect on the flora produced in the intestine.

9 cl, 1 dwg, 3 tbl, 10 ex

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RU 2 527 769 C2

Authors

Kristian Khubshverlen

Khans Lokher

Dates

2014-09-10Published

2009-05-08Filed