PHARMACEUTICAL COMBINATIONS CONTAINING PYRIDO[4,3-d]PYRIMIDINE DERIVATIVES AS HSP90 INHIBITOR AND HER2 INHIBITOR Russian patent published in 2014 - IPC A61K31/422 A61K39/395 A61P35/00 

Abstract RU 2532375 C2

FIELD: medicine.

SUBSTANCE: invention represents a combination for treating breast cancer, containing the HSP90 inhibitor and HER2 inhibitor, wherein the HSP90 inhibitor represents ethylamide 5-(2,4-dihydroxy-5-isopropylphenyl)-4-(4-morpholin-4-ylmethylphenyl)isoxazole-3-carboxylic acid or its pharmaceutically acceptable salt, as well as a method of treating breast cancer, which involves administering an effective amount of this combination in a patient in need thereof.

EFFECT: combination possesses the higher effectiveness as compared to its individual ingredients.

6 cl, 1 ex, 1 tbl, 1 dwg

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RU 2 532 375 C2

Authors

Karlos Garsija-Ehcheverrija

Mikaehl' Jensen

Dates

2014-11-10Published

2009-11-25Filed