ENANTIOMERS OF SPIRO-OXINDOLE COMPOUNDS AND USING THEM AS THERAPEUTIC AGENTS Russian patent published in 2014 - IPC C07D491/20 A61K31/404 A61P21/00 A61P23/00 A61P29/00 

Abstract RU 2535667 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to a new compound, namely to (S)-enantiomer of 1'-{[5-(trifluoromethyl)furan-2-yl]methyl}spiro[furo[2,3-f][1,3]benzodioxol-7,3'-indole]-2'(1'H)-one of formula (I), and a method for preparing it which is effective for treating diseases and conditions, such as pain, an intensity of which can be reduced or relieved by modulating potential-dependent sodium channel gatings.

EFFECT: invention refers to the pharmaceutical composition of the above compound, methods of treating and a method of relieving an ion flux through the potassium channel gating in a cell.

10 cl, 5 tbl, 6 dwg, 11 ex

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RU 2 535 667 C2

Authors

Chafeev Mikhail

Fu Tszjan'Min'

Kad'E Zhan-Zhak

Dates

2014-12-20Published

2010-06-28Filed