ANTITUBERCULOUS THERAPEUTIC AGENT: COMPOSITION OF IMIDAZO[1,2-b]TETRAZINE AND PYRAZINAMIDE Russian patent published in 2015 - IPC C07D487/04 C07D403/04 A61K31/395 A61P31/06 

Abstract RU 2545458 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to a chemical compound of formula wherein R=benzyl and to an antituberculous therapeutic agent representing a composition of imidazo[1,2-b][1,2,4,5]tetrazine derivative of formula I, wherein R=benzyl, isopropyl or phenyl and the known antituberculous preparation pyrazinamide with the ingredients in mole ratio 1:1.

EFFECT: there are prepared new antituberculous therapeutic agents.

2 cl, 2 tbl, 6 ex

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RU 2 545 458 C2

Authors

Bekker Ol'Ga Borisovna

Danilenko Valerij Nikolaevich

Ishmetova Rashida Irshotovna

Korotina Anna Vladimirovna

Maslov Dmitrij Antonovich

Rusinov Gennadij Leonidovich

Tolshchina Svetlana Gennad'Evna

Charushin Valerij Nikolaevich

Dates

2015-03-27Published

2013-08-01Filed