6-SUBSTITUTED 3-AZOLYLIMIDAZO[1,2-b][1,2,4,5]TETRAZINES SHOWING ANTICANCER ACTIVITY Russian patent published in 2014 - IPC C07D487/04 A61K31/395 A61P35/00 

Abstract RU 2527258 C1

FIELD: chemistry.

SUBSTANCE: there are described new derivatives of imidazo[1,2-b][1,2,4,5]tetrazines of general formula (I) wherein: Het=4-methylimidazol-1-yl, R=H or Het=3,5-dimethylpyrazol-1-yl, R=propylthio, and based anticancer agents for treating oncological patients.

EFFECT: higher clinical effectiveness.

2 cl, 1 tbl, 2 ex

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RU 2 527 258 C1

Authors

Bekker Ol'Ga Borisovna

Danilenko Valerij Nikolaevich

Ignatenko Nina Konstantinovna

Ishmetova Rashida Irshotovna

Rusinov Gennadij Leonidovich

Tolshchina Svetlana Gennad'Evna

Charushin Valerij Nikolaevich

Shtil' Aleksandr Al'Bertovich

Dates

2014-08-27Published

2013-02-19Filed