2-[(2-METHYLPHENYL)IMINO]-9-OXO-7-PHENYL-8-(3-PHENYL-2-QUINOXALINYL)-1,6-DIOXASPIRO[4,4]-NONE-3,7-DIENE-3,4-DICARBOXYLIC ACID DIMETHYL ESTER SHOWING ANTINOCICEPTIVE ACTIVITY AND METHOD FOR PRODUCING IT Russian patent published in 2015 - IPC C07D493/10 A61K31/343 A61P29/00 

Abstract RU 2556995 C2

FIELD: chemistry.

SUBSTANCE: invention refers to a new compound, namely to 2-[(2-methylphenyl)imino]-9-oxo-7-phenyl-8-(3-phenyl-2-quinoxalinyl)-1,6-dioxaspiro[4,4]none-3,7-diene-3,4-dicarboxylic acid dimethyl ester of formula possessing antinociceptive activity, and a method for producing it consisting in synthesis of 4-(3-phenylquinoxalin-2-yl)-5-phenylfurane-2,3-dione, acetylene dicarboxylic acid dimethyl ester and o-methylphenylisonitrile.

EFFECT: preparing the new compound.

2 cl, 1 tbl, 4 ex

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RU 2 556 995 C2

Authors

Lisovenko Natal'Ja Jur'Evna

Makhmudov Ramiz Ragibovich

Drjakhlov Artem Vasil'Evich

Dates

2015-07-20Published

2013-07-30Filed