NEW POLYMORPH Russian patent published in 2015 - IPC C07D403/12 A61K31/4025 A61P13/02 

Abstract RU 2559633 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to a new polymorph, namely to a solid form of 1-(2-methyl-4-(2,3,4,5-tetrahydro-1-benzazepin-1-ylcarbonyl)benzylcarbamoyl)-L-proline-N,N-dimethylamine, pharmaceutical compositions containing them.

EFFECT: producing the pharmaceutical compositions for treating a disease or a condition mediated by V2 vasopressin receptors.

10 cl, 14 tbl, 12 dwg

Similar patents RU2559633C2

Title Year Author Number
METHOD OF PRODUCING 1-(2-METHYL-4-(2,3,4,5-TETRAHYDRO-1-BENZAZEPIN-1-YLCARBONYL)BENZYLCARBAMOYL)-L-PROLINE-N,N-DIMETHYLAMIDE 2012
  • Pil Valeri Elizabet
RU2594164C2
CONDENSED AZEPINES, PHARMACEUTICAL COMPOSITION COMPRISING THEREOF, METHOD FOR TREATMENT BY USING INDICATED COMPOSITION 2001
  • Ashuehrt Dorin Mehri
  • Pitt Gari Robert Uil'Jam
  • Khadson Piter
  • Jej Kristofer Martin
  • Franklin Richard Dzheremi
RU2259367C2
CONDENSED AZEPINE DERIVATIVES AS ANTIDIUTETIC AGENTS 2001
  • Ehshuehrt Dorin Mehri
  • Pitt Gari Robert Uil'Jam
  • Khadson Piter
  • Jej Kristofer Martin
  • Franklin Richard Dzheremi
  • Sempl Grem
  • Dzhenkins Dehvid Pol
RU2269517C2
CRYSTALLINE FORMS OF THE TLR7/TLR8 INHIBITOR 2019
  • Bieri, Nicole
  • Kordikowski, Andreas
  • Li, Bin
  • Lustenberger, Philipp
  • Ramos, Rita
  • Sethuraman, Vijay
  • Zhang, Sisi
RU2792005C2
COCRYSTALLINE FORM OF 2,8-DIMETHYL-5-PHENETHYL-2,3,4,5-TETRAHYDRO-1H-PYRIDO[4,3-b]INDOLE 2022
  • Kravchenko Dmitrii Vladimirovich
  • Dmitrieva Irina Gennadevna
RU2806046C1
BICYCLIC AGONISTS OF VASOPRESSIN 2000
  • Ashuehrt Dorin Mehri
  • Pitt Gari Robert Uil'Jam
  • Khadson Piter
  • Jej Kristofer Martin
  • Franklin Richard Dzheremi
RU2254332C2
NOVEL SOLID FORMS (2S,3S,4S,5R,6S)-3,4,5-TRIHYDROXY-6-(((4AR,10AR)-7-HYDROXY-1-PROPYL-1,2,3,4,4A,5,10,10A-OCTAHYDROBENZO[G]QUINOLIN-6-YL)OXY)TETRAHYDRO-2H-PYRAN-2-CARBOXYLIC ACID 2020
  • Jensen, Klaus, Gervig
  • Jorgensen, Morten
  • Dzhukhl, Martin
  • Kvaerno, Lisbet
  • De Diego, Khejdi, Lopez
  • Fredkholt, Karin
  • Terkelsen, Frans Dennis
  • Frikhed, Tobias Gilling
  • Yakobsen, Mikkel Fog
RU2820501C2
CONDENSED BENZAZEPINE DERIVATIVE, AN INTERMEDIATE COMPOUND FOR ITS SYNTHESIS, A PHARMACEUTICAL COMPOSITION 1994
  • Akikhiro Tanaka
  • Khirojuki Kosio
  • Nobuaki Taniguti
  • Akira Matsukhisa
  • Ken-Itiro Sakamoto
  • Atsuki Jamazaki
  • Takejuki Jatsu
RU2129123C1
NOVEL CRYSTALLINE FORMS OF SODIUM SALT OF (4-{4-[5-(6-TRIFLUOROMETHYL-PYRIDIN-3-YLAMINO)PYRIDIN-2-YL]PHENYL}CYCLOHEXYL) ACETIC ACID 2011
RU2612556C2
CRYSTALLINE FORM OF METHYL ESTER 3-(N-P-TOLYLACETAMIDO) METHYL)-2,3,4,5-TETRAHYDROBENZO[f][1,4]OXAZEPINE-4-CARBOXAMIDE)THIOPHENE-2-CARBOXYLIC ACID, ACTIVE COMPONENT, PHARMACEUTICAL COMPOSITION AND DRUG 2014
  • Leonov Sergej Viktorovich
  • Marusich Elena Ivanovna
RU2594154C2

RU 2 559 633 C2

Authors

Chell'Strem Jokhan Khenrik

Jokhanson B'Ern Ehrik

Vil'Khel'Msen Tomas

Dates

2015-08-10Published

2011-03-31Filed