OBTAINING 13-CYCLOHEXYL-3-METHOXY-6-[METHYL-(2-{ 2-[METHYL-(SULPHAMOYL)-AMINO]-ETHOXY}-ETHYL)-CARBAMOYL]-7H-INDOLO-[2,1-α]-[2]-BENZAZEPIN-10-CARBOXYLIC ACID Russian patent published in 2015 - IPC C07D223/14 C07C307/06 C07D487/04 

Abstract RU 2559886 C2

FIELD: chemistry.

SUBSTANCE: present invention relates to a method of producing 13-cyclohexyl-3-methoxy-6-[methyl-(2-{2-[methyl-(sulphamoyl)-amino]-ethoxy}-ethyl)-carbamoyl]-7H-indolo-[2,1-α]-[2]-benzazepin-10-carboxylic acid and a novel compound used in the method, and specifically to tert-butyl(methyl-{2-[2-(methylamino)-ethoxy]-ethyl}-sulphamoyl)-carbamate.

EFFECT: method is easier to implement and is more efficient than the existing method.

8 cl, 5 ex

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Authors

Govarts Tom Kornelis Khortense

Bongartz Zhan-P'Er Andre Mark

Niste Patrik Khubert J.

Dates

2015-08-20Published

2011-06-24Filed