CARBAMYLATED DARBEPOETIN 9C-DEPO, METHOD FOR PRODUCTION THEREOF AND USE THEREOF AS MEDICINAL AGENT HAVING CYTOPROTECTIVE ACTION Russian patent published in 2016 - IPC A61K38/16 C07K14/505 

Abstract RU 2575773 C2

FIELD: chemistry.

SUBSTANCE: group of inventions discloses a method of producing carbamylated darbepoetin 9C-DEPO, which is carbamylated on all amino acid residues of lysine which are part of a darbepoetin molecule, containing a carbamylated amino acid residue of alanine in the N-terminal region of said protein, which includes carbamylation of darbepoetin in the presence of cyanates, as well as a medicinal agent which includes carbamylated darbepoetin 9C-DEPO.

EFFECT: group of inventions has marked cytoprotective action.

2 cl, 3 dwg, 3 ex

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RU 2 575 773 C2

Authors

Shukurov Rakhim Rakhmankulyevich

Khamitov Ravil' Avgatovich

Krjazhevskikh Irina Sergeevna

Dates

2016-02-20Published

2013-07-09Filed