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2 445 310

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IPC

C07D417/14(2006-01-01)

A61K31/541(2006-01-01)

A61K31/549(2006-01-01)

A61P7/02(2006-01-01)

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Application

2010114404/04, 2010-04-12

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Start date

2010-04-12

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Actual filing date

2010-04-12

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Published

2012-03-20

(72)

Inventor

Chupakhin Oleg NikolaevichSidorova Larisa PetrovnaPerova Natal'Ja MikhajlovnaRusinov Vladimir LeonidovichMakarov Vladimir AleksandrovichVasil'Eva Tat'Jana Mikhajlovna

(73)

Holder

Federal'Noe Gosudarstvennoe Avtonomnoe Obrazovatel'Noe Uchrezhdenie Vysshego Professional'Nogo Obrazovanija Federal'Nyj Universitet Imeni Pervogo Prezidenta Rossii B.N. El'Tsina"

2-PIPERIDINO-5-(THIENYL-2)- AND 2-PIPERIDINO-5-(THIENYL-3)- 6H-1,3,4-THIADIAZINES HYDROBROMIDES POSSESSING ANTIAGGREGANT ACTION Russian patent published in 2012 - IPC C07D417/14 A61K31/541 A61K31/549 A61P7/02

Abstract RU 2445310 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention refers to 2-piperidino-5-(thienyl-2)-6H-1,3,4-thiadiazines, hydrobromides (of general formula I) and 2-piperidino-5-(thienyl-3)-6H-1,3,4-thiadiazines, hydrobromides (of general formula II) which possess antiaggregant action. wherein R=H; Cl; Br R₁=H; Cl.

EFFECT: given compounds may be used for preparing cardiologic drugs and enable better treatment of various cardiovascular diseases, including myocardial infarction and thrombotic apoplexy.

1 cl, 2 tbl, 5 ex

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RU 2 445 310 C2

Authors

Chupakhin Oleg Nikolaevich

Sidorova Larisa Petrovna

Perova Natal'Ja Mikhajlovna

Rusinov Vladimir Leonidovich

Makarov Vladimir Aleksandrovich

Vasil'Eva Tat'Jana Mikhajlovna

Dates

2012-03-20—Published

2010-04-12—Filed