TETRACYCLIC COMPOUNDS Russian patent published in 2016 - IPC C07D209/88 C07D307/92 C07D333/76 C07D401/06 C07D405/12 C07D471/04 C07D491/107 A61K31/403 A61K31/343 A61P35/00 

Abstract RU 2585622 C2

FIELD: organic chemistry.

SUBSTANCE: invention relates to organic chemistry, specifically to a particular 9-ethyl-6,6-dimethyl-8-(4-morpholine-4-yl-piperidine-1-yl)-11-oxo-6,11-dihydro-5H-dihydro-5H-benzo [b]carbazole-3-carbonitrile . Invention also relates to a medicament, an ALK inhibitor and pharmaceutical composition based on particular benzo-carbazole derivative.

EFFECT: novel benzo-carbazole derivatives which are useful in treating cancer are obtained.

7 cl, 49 tbl, 1218 ex

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RU 2 585 622 C2

Authors

Kinosita Kazutomo

Asokh Kokhsuke

Furuiti Noriyuki

Ito Tosiya

Kavada Khatsuo

Isii Nobuya

Sakamoto Khirosi

Khong Voosang

Park Mindzeong

Ono Esiyuki

Kato Yasukharu

Morikami Kendzi

Emura Takasi

Oikava Nobukhiro

Dates

2016-05-27Published

2010-06-09Filed