FIELD: medicine; pharmaceuticals.
SUBSTANCE: invention relates to a novel sulphonamide compound of formula (I) having inhibiting ribonucleotide reductase activity, and to pharmaceutical compositions containing it as an active ingredient.
[Formula 1]
EFFECT: obtaining novel compounds having ribonucleotide reductase inhibitory activity, which can be used as an antitumour agent, where the tumor is selected from a group, consisting of breast cancer, stomach cancer, lung cancer, pancreatic cancer, Ewing's sarcoma, glioblastoma, liver cancer, mesothelioma, prostate cancer, ovarian cancer, kidney cancer, colon and rectal cancer, melanoma and blood cancer.
31 cl, 4 dwg, 21 tbl, 354 ex
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Authors
Dates
2020-09-21—Published
2017-05-30—Filed