DIOXINO- AND OXAZIN-[2,3-D]PYRIMIDINE COMPOUNDS AS PHOSPHOINOSITIDE 3-KINASE INHIBITORS AND METHODS FOR USE THEREOF Russian patent published in 2017 - IPC C07D491/04 C07D491/56 A61K31/519 A61P35/00 A61P29/00

Abstract RU 2612251 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a compound of formula I , which are used as inhibitors of phosphoinositide 3-kinase (PI3-kinase), having anticancer activity, anti-inflammatory activity or immunoregulatory properties.

EFFECT: technical result is obtaining novel compounds of formula I, as well as pharmaceutical compositions based thereon, which can be used for producing a drug for treating cancer, in particular, cerebral cancer.

23 cl, 1 tbl, 41 ex

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Authors

Dates

2017-03-03—Published

2013-08-29—Filed