NEW REBAMIPIDE PRODRUGS, METHOD FOR THEIR PREPARATION AND APPLICATION Russian patent published in 2017 - IPC C07D215/227 A61K31/4704 A61P1/04 

Abstract RU 2612509 C2

FIELD: biotechnology.

SUBSTANCE: invention relates to a compound of formula 1

that is a new rebamipide prodrug, and to the pharmaceutical composition thereof.

EFFECT: new rebamipide prodrug with absorption rate 25 times higher than that of rebamipide, which can be used for prevention or treatment of gastric ulcer, acute gastritis, chronic gastritis, xerophthalmia, cancer, osteoarthritis, rheumatoid arthritis, or obesity.

7 cl, 3 tbl, 204 ex, 1 dwg

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RU 2 612 509 C2

Authors

Dates

2017-03-09Published

2013-06-26Filed