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2 629 999

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(51)

IPC

C07D471/04(2006-01-01)

A61K31/416(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2012150759, 2012-11-28

(24)

Start date

2006-06-21

(22)

Actual filing date

2012-11-28

(45)

Published

2017-09-05

(72)

Inventor

Ibrahim Prahbha N.Artis Dean R.Bremer RyanMamo ShumeyeNespi MarikaZhang ChaoZhang JiazhongZhu Yong-LiangTsai JamesHirth Klaus-PeterBollag GideonSpevak WayneCho HannaGillette Samuel J.Vu GuoksiamZhu KhongyaoShi Shengkhua

(73)

Holder

Plexxikon, Inc.

PYROLLO [2,3-B]PYRIDINE DERIVATIVES AS PROTEIN KINASE INHIBITORS Russian patent published in 2017 - IPC C07D471/04 A61K31/416 A61P35/00

Abstract RU 2629999 C2

FIELD: pharmacology.

SUBSTANCE: invention relates to a compound of formula

which exhibits activity against protein kinases, as well as to methods of its preparation and pharmaceutical compositions.

EFFECT: increased compound activity.

15 cl, 8 tbl, 9 ex

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RU 2 629 999 C2

Authors

Ibrahim Prahbha N.

Artis Dean R.

Bremer Ryan

Mamo Shumeye

Nespi Marika

Zhang Chao

Zhang Jiazhong

Zhu Yong-Liang

Tsai James

Hirth Klaus-Peter

Bollag Gideon

Spevak Wayne

Cho Hanna

Gillette Samuel J.

Vu Guoksiam

Zhu Khongyao

Shi Shengkhua

Dates

2017-09-05—Published

2012-11-28—Filed