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2 632 885

(13)

(51)

IPC

C07D213/82(2006-01-01)

C07D401/12(2006-01-01)

C07D405/14(2006-01-01)

A61K31/444(2006-01-01)

A61K31/4545(2006-01-01)

A61P35/00(2006-01-01)

A61P43/00(2006-01-01)

(21) (22)

Application

2014135401, 2013-01-30

(24)

Start date

2013-01-30

(22)

Actual filing date

2013-01-30

(45)

Published

2017-10-11

(72)

Inventor

Okhki KhitosiOta MasakhiroTakeuti KosukeVatanabe KhideakiYamaguti AkitakeSibata JosikhiroTominaga YuitiDzimbo TakesiKobayasi KejdziroKobayasi KatsukhiroFukatsu Dajsuke

(73)

Holder

Dajiti Sankio Kompani, Limited

PYRIDON DERIVATIVES Russian patent published in 2017 - IPC C07D213/82 C07D401/12 C07D405/14 A61K31/444 A61K31/4545 A61P35/00 A61P43/00

Abstract RU 2632885 C2

FIELD: pharmacology.

SUBSTANCE: invention relates to compounds of formula (I)

New compounds and their crystalline forms that inhibit Ax1 and are useful for treatment of diseases caused by Ax1 hyperfunction, diseases associated with Ax1 hyperfunction, and/or diseases accompanied by Ax1 hyperfunction, such as hyperoproliferative disease.

EFFECT: means have increased effectiveness.

37 cl, 16 tbl, 107 ex, 16 dwg

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RU 2 632 885 C2

Authors

Okhki Khitosi

Ota Masakhiro

Takeuti Kosuke

Vatanabe Khideaki

Yamaguti Akitake

Sibata Josikhiro

Tominaga Yuiti

Dzimbo Takesi

Kobayasi Kejdziro

Kobayasi Katsukhiro

Fukatsu Dajsuke

Dates

2017-10-11—Published

2013-01-30—Filed