(N-SUBSTITUTED IMIDAZOLE)-CARBOXYLIC ESTER CHIRAL COMPOUND CONTAINING ETHER SIDE CHAIN, PREPARATION METHOD AND APPLICATION Russian patent published in 2018 - IPC C07D233/90 A61K31/4174 A61P23/00 A61P25/20 

Abstract RU 2659784 C2

FIELD: chemistry.

SUBSTANCE: invention relates to organic chemistry, in particular to an (N-substituted imidazole)-carboxylic acid ester chiral compound containing an ether side chain of formula (I) and a pharmaceutically acceptable salt thereof. Invention also relates to a process for the preparation of a compound of formula (I), a pharmaceutically acceptable salt thereof and use thereof.

EFFECT: technical result: an ester chiral compound is obtained useful in the preparation of drugs inhibiting the central nervous system, which can cause sedative, hypnotic and/or anesthetic effects.

9 cl, 3 dwg, 4 tbl, 11 ex

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RU 2 659 784 C2

Authors

Chzhan Venshen

Yan Tszyun

Lyu Tszin

Tan Lej

Ke Boven

Dates

2018-07-04Published

2014-10-30Filed