FIELD: chemistry.
SUBSTANCE: present invention relates to a compound of formula I, or a pharmaceutically acceptable salt thereof.
formula.
In formula IX and Y are selected from any of following 1) or 2): 1) X is C = O, Y is NH; 2) X is C = O, Y is absent; R is selected from any of the following groups: C1-C25 alkyl group which is unsubstituted or substituted with halogen, an ester group, amino acid derivatives; unsubstituted C3-C25 cycloalkyl group; a phenyl ring unsubstituted or substituted with an ester group, halogen; unsubstituted naphthalic ring; pyridine ring, unsubstituted or substituted with halogen; pyridazine ring substituted with halogen; unsubstituted indole ring; unsubstituted C2-C25 alkenyl or alkynyl group.
EFFECT: invention is capable of slow release of 2-tert-butyl-4-methoxyphenol in vivo and is able to maintain stable concentration of 2-tert-butyl-4-methoxyphenol in blood plasma.
8 cl, 4 dwg, 3 tbl, 71 ex
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Authors
Dates
2019-12-09—Published
2017-02-22—Filed