FIELD: chemistry.
SUBSTANCE: present invention relates to a compound of formula (I):
,
optionally linked with an effector moiety, where the effector moiety includes an effector that is a diagnostically active nuclide or a therapeutically active nuclide.
EFFECT: obtaining novel compounds of formula (I), as well as pharmaceutical compositions based thereon, which inhibit the activity of the NTR1 ligand.
26 cl, 30 ex, 9 dwg
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