NEUROTENSIN RECEPTOR LIGANDS Russian patent published in 2018 - IPC C07D231/14 A61K31/415 A61P35/00 

Abstract RU 2671970 C2

FIELD: chemistry.

SUBSTANCE: present invention relates to a compound of formula (I):

,

optionally linked with an effector moiety, where the effector moiety includes an effector that is a diagnostically active nuclide or a therapeutically active nuclide.

EFFECT: obtaining novel compounds of formula (I), as well as pharmaceutical compositions based thereon, which inhibit the activity of the NTR1 ligand.

26 cl, 30 ex, 9 dwg

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RU 2 671 970 C2

Authors

Osterkamp Frank

Smerling Kristiane

Rajneke Ulrikh

Khaaze Kristian

Ungeviss Yan

Dates

2018-11-08Published

2013-12-06Filed