FIELD: chemistry.
SUBSTANCE: present invention relates to a compound of formula (I):
,
optionally linked with an effector moiety, where the effector moiety includes an effector that is a diagnostically active nuclide or a therapeutically active nuclide.
EFFECT: obtaining novel compounds of formula (I), as well as pharmaceutical compositions based thereon, which inhibit the activity of the NTR1 ligand.
26 cl, 30 ex, 9 dwg
Title | Year | Author | Number |
---|---|---|---|
A CONJUGATE CONTAINING A NEUROTENSIN RECEPTOR LIGAND AND ITS APPLICATION | 2015 |
|
RU2743781C2 |
COMPLEX CONTAINING A PSMA-TARGETING COMPOUND BOUND TO A LEAD OR THORIUM RADIONUCLIDE | 2018 |
|
RU2795398C2 |
BOMBESIN ANALOGUE PEPTIDE ANTAGONIST CONJUGATES | 2009 |
|
RU2523531C2 |
DIAGNOSIS, TREATMENT AND PREVENTION OF CONDITIONS ASSOCIATED WITH THE NEUROTENSIN RECEPTOR | 2017 |
|
RU2796538C2 |
PARAMINOHYPURIC ACID (PAH) AS A KIDNEY PROTECTOR | 2020 |
|
RU2804349C2 |
NOVEL RADIOIMMUNOCONJUGATES AND THEIR APPLICATIONS | 2011 |
|
RU2560587C9 |
NOVEL RADIOIMMUNOCONJUGATES AND USE THEREOF | 2011 |
|
RU2664475C1 |
NEW PSA-BINDING AGENTS AND THEIR USE | 2018 |
|
RU2787105C2 |
PSMA LIGANDS FOR IMAGING AND ENDORADIOTHERAPY | 2018 |
|
RU2807076C2 |
IMMUNOTHERAPY OF MALIGNANT DISEASES OF B-CELLS AND AUTOIMMUNE DISEASES WITH APPLICATION OF CONJUGATE AND NONCONJUGATE ANTIBODIES, COMBINATIONS OF ANTIBODIES AND CONJOINT PROTEINS | 2003 |
|
RU2335297C2 |
Authors
Dates
2018-11-08—Published
2013-12-06—Filed