USE OF THE BISAMIDE MALONIC ACID DERIVATIVE FOR TREATING ALLERGIC AND OTHER HUMAN AND ANIMAL DISEASES Russian patent published in 2019 - IPC C07D403/12 A61K31/4178 A61P11/00 A61P37/00 

Abstract RU 2685277 C1

FIELD: medicine; pharmaceuticals.

SUBSTANCE: invention describes the use of compound 1 or its pharmaceutically acceptable salt, hydrate or solvate as a histamine receptor antagonist of the third type. Also disclosed are a pharmaceutical composition containing compound 1, methods for preventing and/or treating a disorder associated with histamine receptor activity of the third type, and using the compound of formula 1.

(1).

EFFECT: obtaining an effective histamine receptor antagonist of the third type, characterized by high activity and pharmacokinetic characteristics, allowing to use compound 1 when used for therapy of allergic diseases.

12 cl, 8 tbl, 6 ex

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RU 2 685 277 C1

Authors

Nebolsin Vladimir Evgenevich

Dates

2019-04-17Published

2018-05-24Filed