3'-AROYL-1-BENZYL-4'-HYDROXY-1'-(2-HYDROXYETHYL)-6,6-DIMETHYL-6,7-DIHYDROSPIRO[INDOLO-3,2'-PYRROLE]-2,4,5'(1H,1'H,5H)-TRIONES POSSESSING ANALGESIC ACTIVITY AND A METHOD FOR THEIR PREPARATION Russian patent published in 2019 - IPC C07D487/10 A61K31/40 A61P29/00 

Abstract RU 2688931 C1

FIELD: chemistry.

SUBSTANCE: invention relates to organic chemistry and specifically to 3'-aroyl-1-benzyl-4'-hydroxy-1'-(2-hydroxyethyl)-6,6-dimethyl-6,7-dihydrospiro[indolo-3,2'-pyrrole]-2,4,5'(1H,1'H,5H)-triones and a method for production thereof.

.

EFFECT: compounds have analgesic activity.

4 cl, 1 tbl, 3 ex

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RU 2 688 931 C1

Authors

Tretyakov Nikita Alekseevich

Maslivets Andrej Nikolaevich

Makhmudov Ramiz Ragibovich

Galeev Andrej Ruslanovich

Dates

2019-05-23Published

2018-11-15Filed