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2 702 648

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IPC

C07D215/18(2006-01-01)

A61K31/47(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2019121680, 2019-07-11

(24)

Start date

2019-07-11

(22)

Actual filing date

2019-07-11

(45)

Published

2019-10-09

(72)

Inventor

Saiapin Iurii AnatolevichGusakov Evgenii AleksandrovichMazitova Aleksandra MaratovnaTopchu Iuliia AlekseevnaDorogan Igor ViktorovichBumber Ianis AlekseevichMinkin Vladimir Isaakovich

(73)

Holder

Federalnoe Gosudarstvennoe Avtonomnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovaniia Federalnyi Universitet»

5,7-DI(TERT-BUTYL)-2-(4,7-DICHLORO-8-METHYL-5-NITROQUINOLIN-2-YL)-4-NITRO-1,3-TROPOLONE, HAVING CYTOTOXIC ACTIVITY Russian patent published in 2019 - IPC C07D215/18 A61K31/47 A61P35/00

Abstract RU 2702648 C1

FIELD: chemistry.

SUBSTANCE: invention relates to organic chemistry and specifically to 5,7-di(tert-butyl)-2-(4,7-dichloro-8-methyl-5-nitroquinolin-2-yl)-4-nitro-1,3-tropolone of formula 1. 1.

EFFECT: obtaining a novel heterocyclic compound having cytotoxic activity on ovarian cancer cell lines, lung cancer, colon cancer and pancreatic cancer.

1 cl, 1 tbl, 1 ex

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RU 2 702 648 C1

Authors

Saiapin Iurii Anatolevich

Gusakov Evgenii Aleksandrovich

Mazitova Aleksandra Maratovna

Topchu Iuliia Alekseevna

Dorogan Igor Viktorovich

Bumber Ianis Alekseevich

Minkin Vladimir Isaakovich

Dates

2019-10-09—Published

2019-07-11—Filed