FIELD: medicine.
SUBSTANCE: invention relates to compounds characterized by high antibacterial activity of general formula (I), where R1-R2 have values given in description. Invention also relates to pharmaceutical compositions containing said compounds, and to use of said compounds for treating and/or preventing infectious diseases, including those caused by antibiotic-resistant pathogens (including multiresistant strains), in particular, staphylococcal aetiology, e.g. infectious diseases of skin and/or soft tissues, pneumonia, endocarditis or osteomyelitis.
EFFECT: proposed is use of 6-fluoro-3-triazenone indoles for therapy of MRSA-induced infections.
14 cl, 1 dwg, 5 tbl, 1 ex
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