PYRIDOPYRIMIDINONES AND USE THEREOF AS MODULATORS OF N-METHYL-D-ASPARTATE RECEPTOR Russian patent published in 2020 - IPC A61K31/517 A61K31/519 A61P21/00 A61P25/00 A61P25/02 A61P25/04 A61P25/08 A61P25/14 A61P25/16 A61P25/18 A61P25/24 A61P25/28 A61P25/30 A61P29/00 A61P43/00 A61P9/00 A61P9/10 A61P25/22 C07D471/04 

Abstract RU 2717665 C2

FIELD: medicine; pharmaceuticals.

SUBSTANCE: invention relates to a compound of formula I, as well as to a pharmaceutical composition for treating a disease or medical condition mediated by N2RA activity, comprising an effective amount of a compound of formula I and a pharmaceutically acceptable carrier.

EFFECT: disclosed are pyridopyrimidinones and use thereof as n-methyl-d-aspartate receptor modulators.

22 cl, 1 tbl, 1 ex

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RU 2 717 665 C2

Authors

Volgraf Metyu

Tszyan Yu

Villemur Eliziya

Sellers Bendzhamin

U Goshen

Lu Ajtszyun

Dates

2020-03-24Published

2016-04-12Filed