METHOD OF PRODUCING MONOCHLOROACETATES OF SUBSTITUTED 5-, 6-, 7-AMINOINDOLES, HAVING ANTIMICROBIAL ACTION Russian patent published in 2020 - IPC C07D209/40 

Abstract RU 2724605 C1

FIELD: chemistry.

SUBSTANCE: invention relates to a method of producing monochloroacetates of substituted 5-, 6-, 7-aminoindoles, which involves reacting corresponding substituted 5-, 6-, 7-aminoindoles in benzene heated with boiling with monochloroacetic acid.

EFFECT: obtained novel salts, such as 2,3-dimethyl-1H-indole-5-ammonium monochloroacetate, 1,2,3-trimethyl-1H-indole-5-ammonium monochloroacetate, 2,3-dimethyl-5-methoxy-1H-indole-6-ammonium monochloroacetate, 5-methoxy-1,2,3-trimethyl-1H-indole-6-ammonium monochloroacetate, 2,3-dimethyl-1H-indole-7-ammonium monochloroacetate and 1,2,3-trimethyl-1H-indole-5-ammonium monochloroacetate, can be used as water-soluble synthetic antimicrobial preparations.

1 cl, 6 ex

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RU 2 724 605 C1

Authors

Stepanenko Irina Semenovna

Yamashkin Semen Aleksandrovich

Batarsheva Alena Aleksandrovna

Slastnikov Evgenij Dmitrievich

Dates

2020-06-25Published

2019-08-09Filed