CHEMICAL SYNTHESIS AND ANTI-TUMOR AND ANTI-METASTATIC EFFECTS OF CONJUGATE OF DOUBLE ACTION Russian patent published in 2020 - IPC C07D305/14 C07D405/12 C07D409/12 C07K5/37 A61K31/337 A61K47/54 A61K47/65 A61P35/00 A61P35/04 

Abstract RU 2729419 C2

FIELD: pharmaceuticals.

SUBSTANCE: present invention provides chemical synthesis, anti-tumor and anti-metastatic effects of a double-action conjugate presented by formula I.

EFFECT: synthesis of the conjugate of formula I is carried out by a combination of solid-phase and liquid-phase synthesis, and said conjugate can be used for producing antineoplastic drugs, which is confirmed by reliable results of biological studies.

22 cl, 37 dwg, 13 tbl, 43 ex

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RU 2 729 419 C2

Authors

Lyu Gan

Chzhao Nan

Ma Yao

Dates

2020-08-06Published

2011-05-27Filed