METHODS OF USING AGONISTS FXR Russian patent published in 2020 - IPC A61K31/46 A61K31/4748 A61P1/16 

Abstract RU 2737324 C2

FIELD: medicine.

SUBSTANCE: group of inventions can be used for treating or preventing primary biliary cholangitis in a patient. For this purpose, in the manufacture of a medicament, compound 2-[(1R,3r,5S)-3-({5-cyclopropyl-3-[2-(trifluoromethoxy)phenyl]-1,2-oxazol-4-yl}methoxy)-8-azabicyclo[3.2.1]octan-8-yl]-4-fluoro-1,3-benzothiazole-6-carboxylic acid. Said compound is administered in dose of 10 mcg. Also disclosed are application of said agent in doses of 30 mcg, 60 mcg, 90 mcg, 100 mcg.

EFFECT: group of inventions provides treating, as well as preventing primary biliary cholangitis in a patient.

5 cl, 5 tbl, 2 dwg, 5 ex

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RU 2 737 324 C2

Authors

Laffitte, Bryan

Badman, Michael

Chen, Jin

Lindgren, Sam

Dates

2020-11-27Published

2017-02-20Filed