FXR AGONISTS APPLICATION METHODS Russian patent published in 2021 - IPC A61K31/46 A61K47/54 A61K31/55 A61K31/4748 A61K31/497 A61K31/506 A61P1/16 A61P43/00 

Abstract RU 2743075 C2

FIELD: non-alcoholic steatohepatitis treatment.

SUBSTANCE: invention relates to 2-[(1R,3r,5S)-3-({5-cyclopropyl-3-[2-(trifluoromethoxy) phenyl]-1,2-oxazole-4-yl}methoxy)-8-azabicyclo[3.2.1]octane-8-yl]-4-fluorine-1,3-benzothiazole-6-carboxylic acid for non-alcoholic steatohepatitis treatment (NASH), where the specified compound should be injected at doses of 10 mcg, 30 mcg, 60 mcg, 90 mcg, 120 mcg.

EFFECT: non-alcoholic steatohepatitis treatment.

5 cl, 5 ex, 5 tbl, 5 dwg

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RU 2 743 075 C2

Authors

Laffitte, Bryan

Badman, Michael

Chen, Jin

Lindgren, Sam

Dates

2021-02-15Published

2017-02-20Filed