NEW Β-LACTAMASE INHIBITORS Russian patent published in 2021 - IPC C07D471/08 A61K31/439 A61P31/04 

Abstract RU 2741963 C2

FIELD: pharmaceuticals.

SUBSTANCE: invention relates to a compound of formula (I), in which X is O, having inhibitor properties β-lactamase, or its pharmaceutically acceptable salts, based pharmaceutical composition, preparing a β-lactamase inhibitor for treating a bacterial infection.

EFFECT: novel inhibitors of β-lactamases are disclosed.

4 cl, 7 tbl, 4 ex

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RU 2 741 963 C2

Authors

Khu, Boyuj

Din, Charlz Z.

Khuan, Chzhigan

Lin, Zhujbin

Syao, Minlyan

Se, Tszinshen

Chen, Shukhuej

Li, Chen

Dates

2021-02-01Published

2017-06-02Filed