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2 753 480

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IPC

C07D207/44(2006-01-01)

A61K31/402(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2020130076, 2020-09-14

(24)

Start date

2020-09-14

(22)

Actual filing date

2020-09-14

(45)

Published

2021-08-17

(72)

Inventor

Igidov Nazim MusabekovichBojchuk Sergej VasilevichZykova Svetlana SergeevnaGalembikova Ajgul RafikovnaAukhadieva Aida MaratovnaBikinieva Firyuza FanisovnaNurgatina Ilmira IlyazovnaGankova Kseniya LeonidovnaShustov Maksim Vadimovich

(73)

Holder

Federalnoe Gosudarstvennoe Byudzhetnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovaniya Gosudarstvennaya Farmatsevticheskaya Akademiya» Ministerstva Zdravookhraneniya Rossijskoj FederatsiiFederalnoe Gosudarstvennoe Byudzhetnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovaniya Gosudarstvennyj Meditsinskij Universitet» Ministerstva Zdravookhraneniya Rossijskoj Federatsii

2-AMINO-1-(4-BROMOPHENYL)-5-(3,3-DIMETHYL-2-OXOBUTYLIDENE)-4-OXO-4,5-DIHYDRO-1H-PYRROL-3-CARBOXAMIDE EXHIBITING CYTOTOXIC ACTIVITY AGAINST HUMAN TUMORAL CELLS Russian patent published in 2021 - IPC C07D207/44 A61K31/402 A61P35/00

Abstract RU 2753480 C1

FIELD: medicine.

SUBSTANCE: invention relates to medicine, specifically to 2-amino-1-(4-bromophenyl)-5-(3,3-dimethyl-2-oxobutylidene)-4-oxo-4,5-dihydro-1H-pyrrol-3-carboxamide by the formula I, exhibiting cytotoxic activity against human tumoral cells, and can be applied in treatment of oncological diseases.

EFFECT: invention can be applied in treatment of oncological diseases.

1 cl, 2 dwg, 1 tbl

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RU 2 753 480 C1

Authors

Igidov Nazim Musabekovich

Bojchuk Sergej Vasilevich

Zykova Svetlana Sergeevna

Galembikova Ajgul Rafikovna

Aukhadieva Aida Maratovna

Bikinieva Firyuza Fanisovna

Nurgatina Ilmira Ilyazovna

Gankova Kseniya Leonidovna

Shustov Maksim Vadimovich

Dates

2021-08-17—Published

2020-09-14—Filed