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2 607 920

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IPC

C07D207/50(2006-01-01)

A61K31/4015(2006-01-01)

A61P35/00(2006-01-01)

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Application

2015120527, 2015-05-29

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Start date

2015-05-29

(22)

Actual filing date

2015-05-29

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Published

2017-01-11

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Inventor

Bojchuk Sergej VasilevichZykova Svetlana SergeevnaGalembikova Ajgul RafikovnaRamazanov Bulat RashitovichIgidov Nazim MusabekovichOdegova Tatyana FedorovnaKiselev Maksim AleksandrovichSemina Irina Ivanovna

(73)

Holder

Gosudarstvennoe Byudzhetnoe Obrazovatelnoe Uchrezhdenie Vysshego Professionalnogo Obrazovaniya Gosudarstvennyj Meditsinskij Universitet" Minzdrava RossiiObshchestvo S Ogranichennoj Otvetstvennostyu

ETHYL ETHERS OF 2-AMINO-1-BENZOYLAMINO-4-OXO-5-(2-OXO-2-ARYL-ETHYLIDENE)-4,5-DIHYDRO-1H-PYRROLIDINE-3-CARBOXYLIC ACIDS, HAVING ANTI-TUMOUR ACTIVITY AND METHOD FOR PRODUCTION THEREOF Russian patent published in 2017 - IPC C07D207/50 A61K31/4015 A61P35/00

Abstract RU 2607920 C2

FIELD: chemistry.

SUBSTANCE: invention relates to novel compounds of general formula Ia-d, where R=CH₃O (Ia), C₂H₅O (Ib), Br (Ic), Cl (Id), which have anticancer activity. Also disclosed is a method of producing compounds of formula Ia-d and their application for producing drug preparations for treating oncological diseases.

EFFECT: compounds exhibit low toxicity.

3 cl, 4 dwg, 1 tbl, 6 ex

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RU 2 607 920 C2

Authors

Bojchuk Sergej Vasilevich

Zykova Svetlana Sergeevna

Galembikova Ajgul Rafikovna

Ramazanov Bulat Rashitovich

Igidov Nazim Musabekovich

Odegova Tatyana Fedorovna

Kiselev Maksim Aleksandrovich

Semina Irina Ivanovna

Dates

2017-01-11—Published

2015-05-29—Filed