QUATERNARY AMMONIUM SALTS OF DIAZAADAMANTANS WITH ACTOPROTECTIVE ACTIVITY Russian patent published in 2021 - IPC C07D471/18 A61K31/529 A61P25/26 A61P43/00 

Abstract RU 2760459 C1

FIELD: pharmacology.

SUBSTANCE: invention relates to the field of medical chemistry and pharmacology, namely to new quaternary ammonium salts, specifically to derivatives of 5,7-dimethyl-1,3-diazaadamantan containing monoterpenoid fragments, general formula 1, including spatial isomers, particularly optically active forms, where X: CO, CH2, C = NOH, and Z can be a halogen or a nitro group having an actoprotective effect.

EFFECT: the actoprotective effect of 5,7-dimethyl-1,3-diazaadamantan derivatives of formula 1.

1 cl, 3 dwg, 3 tbl, 8 ex

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RU 2 760 459 C1

Authors

Suslov Evgenii Vladimirovich

Volcho Konstantin Petrovich

Kotliarova Anastasiia Anatolevna

Pavlova Alla Viktorovna

Ponomarev Konstantin Iurevich

Salakhutdinov Nariman Faridovich

Tolstikova Tatiana Genrikhovna

Dates

2021-11-25Published

2021-04-21Filed