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2 612 875

(13)

(51)

IPC

C12N9/16(2006-01-01)

C07D311/22(2006-01-01)

C07D311/94(2006-01-01)

C07C13/42(2006-01-01)

(21) (22)

Application

2015153696, 2015-12-14

(24)

Start date

2015-12-14

(22)

Actual filing date

2015-12-14

(45)

Published

2017-03-13

(72)

Inventor

(73)

Holder

Federalnoe Gosudarstvennoe Byudzhetnoe Uchrezhdenie Nauki Novosibirskij Institut Organicheskoj Khimii Im. N.N. Vorozhtsova Sibirskogo Otdeleniya Rossijskoj Akademii Nauk So Ran)Federalnoe Gosudarstvennoe Byudzhetnoe Uchrezhdenie Nauki Institut Khimicheskoj Biologii I Fundamentalnoj Meditsiny Sibirskogo Otdeleniya Rossijskoj Akademii Nauk So Ran)

MEANS FOR HUMAN TYROSYL-DNA-PHOSPHODIESTERASE 1 ENZYME INHIBITION Russian patent published in 2017 - IPC C12N9/16 C07D311/22 C07D311/94 C07C13/42

Abstract RU 2612875 C1

FIELD: biotechnology.

SUBSTANCE: means which is a chromenone derivative: I, where n = 1 or 2 or II, developing the ability to inhibit the human tyrosyl-DNA phosphodiesterase 1 enzyme is proposed.

EFFECT: it expands the range of means for human tyrosyl-DNA-phosphodiesterase 1 enzyme inhibitors and can be used for development of anticancer drugs.

1 tbl, 7 ex

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RU 2 612 875 C1

Authors

Dates

2017-03-13—Published

2015-12-14—Filed