DELAYED-RELEASE DELIVERY SYSTEMS CONTAINING TRACELESS LINKERS Russian patent published in 2022 - IPC A61K47/61 A61K47/69 A61K47/50 A61P27/02 

Abstract RU 2772690 C2

FIELD: pharmaceutics.

SUBSTANCE: invention relates to drug delivery systems or to its pharmaceutically acceptable salts that are represented by formulas (XXX), (XXXII), (XXXIV), (XXXVI), (XXXVIII) given in the formula of the invention, in which a drug is a biologically active component containing at least one primary or secondary amino group or ring nitrogen atom in azaheteroaryl ring; and R4 is methyl, ethyl, propyl, isopropyl, 1-methylcyclopropyl or methoxymethyl.

EFFECT: new drug delivery systems are developed that provide delayed release of biologically active components for therapeutically significant applications.

5 cl, 9 dwg, 27 tbl, 10 ex

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RU 2 772 690 C2

Authors

Adams, Christopher M.

April, Myriam

Fazal, Tanzina

Forster, Cornelia Jutta

Hall, Edward Charles

Lee, Cameron Chuck-Munn

Dates

2022-05-24Published

2018-04-19Filed