FIELD: pharmaceuticals.
SUBSTANCE: group of inventions relates to pharmaceutical chemistry and pharmacology, namely, to 4-(3,4-dibromothiophene carbonyl)-10-(2-ethoxyacetyl)-2,6,8,12-tetraacetyl-2,4,6,8,10,12-hexaazatetracyclo[5,5,0,03,11,05,9]dodecane by the formula (I) and to a method for production thereof through acylation of 4-(3,4-dibromothyophene carbonyl)-2,6,8,12-tetraacetyl-2,4,6,8,10,12-hexaazatetracyclo[5,5,0,0 3,11,05,9]dodecane with ethoxyacetyl chloride.
EFFECT: 4-(3,4-dibromothiophene carbonyl)-10-(2-ethoxyacetyl)-2,6,8,12-tetraacetyl-2,4,6,8,10,12-hexaazatetracyclo[5,5,0,03,11,05,9]dodecane exhibiting analgesic activity.
2 cl, 3 tbl, 2 ex
| Title |
Year |
Author |
Number |
| 4,10-DI(ETHOXYACETYL)-2,6,8,12-TETRAACETYL-2,4,6,8,10,12-HEXAAZATETRACYCLO[5,5,0,0,0] DODECANE AS AN ANALGESIC AGENT AND A METHOD FOR PRODUCTION THEREOF |
2020 |
- Krylova Svetlana Gennadevna
- Poveteva Tatyana Nikolaevna
- Suslov Nikolaj Innokentevich
- Zueva Elena Petrovna
- Nesterova Yuliya Vladimirovna
- Afanaseva Olga Gennadevna
- Kulpin Pavel Valerevich
- Amosova Evdokiya Naumovna
- Razina Tatyana Georgievna
- Rybalkina Olga Yurevna
- Safonova Elena Andreevna
- Zhdanov Vadim Vadimovich
- Kalashnikov Aleksandr Ivanovich
- Bajbakova Olga Vladimirovna
- Bakholdina Lyubov Alekseevna
- Eremina Valeriya Valerevna
- Sonina Ekaterina Georgievna
- Kulagina Darya Aleksandrovna
- Sysolyatin Sergej Viktorovich
|
RU2736936C1 |
| 4-(3,4-DIBROMOTHYOPHENE CARBONYL)-2,6,8,10,12-PENTAACETYL-2,4,6,8,10,12 HEXAAZAISOWURTZITANE AS AN ANALGESIC AGENT AND METHOD FOR ITS PREPARATION |
2021 |
- Krylova Svetlana Gennadevna
- Poveteva Tatyana Nikolaevna
- Suslov Nikolaj Innokentevich
- Zueva Elena Petrovna
- Nesterova Yuliya Vladimirovna
- Afanaseva Olga Gennadevna
- Kulpin Pavel Valerevich
- Kiseleva Elena Andreevna
- Amosova Evdokiya Naumovna
- Razina Tatyana Georgievna
- Rybalkina Olga Yurevna
- Safonova Elena Andreevna
- Zhdanov Vadim Vadimovich
- Kalashnikov Aleksandr Ivanovich
- Bajbakova Olga Vladimirovna
- Bakholdina Lyubov Alekseevna
- Eremina Valeriya Valerevna
- Sonina Ekaterina Georgievna
- Kulagina Darya Aleksandrovna
- Sysolyatin Sergej Viktorovich
- Alekseeva Natalya Alekseevna
|
RU2769523C1 |
| 4-(2-ETOXYACETYL)-2,6,8,10,12-PENTAACETYL-2,4,6,8,10,12-HEXAAZATETRACYCLO [5,5,0,0,0] DODECANE AS ANALGETIC AND METHOD OF ITS OBTAINING |
2023 |
- Krylova Svetlana Gennadevna
- Poveteva Tatyana Nikolaevna
- Suslov Nikolaj Innokentevich
- Zueva Elena Petrovna
- Nesterova Yuliya Vladimirovna
- Afanaseva Olga Gennadevna
- Kulpin Pavel Valerevich
- Kiseleva Elena Aleksandrovna
- Rybalkina Olga Yurevna
- Zhdanov Vadim Vadimovich
- Bajbakova Olga Vladimirovna
- Eremina Valeriya Valerevna
- Kulagina Darya Aleksandrovna
- Alekseeva Natalya Alekseevna
- Chikina Majya Viktorovna
- Sysolyatin Sergej Viktorovich
|
RU2808905C1 |
| 4-(3,4-DIBROMOTHIOPHENE CARBONYL)-2,6,8,12-TETRAACETYL-2,4,6,8,10,12-HEXAAZATETRACYCLO[5,5,0,0,0]DODECANE AS ANALGESIC AGENT AND METHOD FOR PRODUCTION THEREOF |
2014 |
- Krylova Svetlana Gennad'Evna
- Amosova Evdokija Naumovna
- Zueva Elena Petrovna
- Razina Tat'Jana Georgievna
- Rybalkina Ol'Ga Jur'Evna
- Lopatina Ksenija Aleksandrovna
- Sysoljatin Sergej Viktorovich
- Kalashnikov Aleksandr Ivanovich
- Malykhin Valerij Viktorovich
- Dygaj Aleksandr Mikhajlovich
- Zhdanov Vadim Vadimovich
- Vorozhtsov Aleksandr Borisovich
- Zhukov Aleksandr Stepanovich
|
RU2565766C1 |
| 4,10-DI(ETOXYACETIL)-2,6,8,12-TETRAACETIL-2,4,6,8,10,12-HEXAAZATETRACYCLO [5,5,0,0,0]DODECANE AS ANTI-INFLAMMATORY |
2022 |
- Krylova Svetlana Gennadevna
- Kiseleva Elena Aleksandrovna
- Poveteva Tatyana Nikolaevna
- Suslov Nikolaj Innokentevich
- Zueva Elena Petrovna
- Amosova Evdokiya Naumovna
- Zhdanov Vadim Vadimovich
- Bajbakova Olga Vladimirovna
- Eremina Valeriya Valerevna
- Kulagina Darya Aleksandrovna
- Sysolyatin Sergej Viktorovich
|
RU2798994C1 |
| 4-(3,4-DIBROMOTHIOPHENE CARBONYL)-2,6,8,12-TETRAACETYL-2,4,6,8,10,12-HEXAAZATETRACYCLO[5,5,0,0,0]DODECANE USED AS AN ANTICONVULSANT |
2018 |
- Krylova Svetlana Gennadevna
- Poveteva Tatyana Nikolaevna
- Sysolyatin Sergej Viktorovich
- Suslov Nikolaj Innokentevich
- Zueva Elena Petrovna
- Nesterova Yuliya Vladimirovna
- Afanaseva Olga Gennadevna
- Lopatina Kseniya Aleksandrovna
- Kulpin Pavel Valerevich
- Zhdanov Vadim Vadimovich
- Kulagina Darya Aleksandrovna
- Malykhin Valerij Viktorovich
- Vorozhtsov Aleksandr Borisovich
|
RU2684107C1 |
| 4,10-BIS((±)-5-BENZOYL-2,3-DIHYDRO-1H-PYRROLO[1,2-A]PYRROLE-1-CARBONYL)-2,6,8,12-TETRAACETYL-2,4,6,8,10,12-HEXAAZATETRACYCLO[5,5,0,0,0]DODECANE AS ANALGETIC MEANS AND METHOD OF ITS OBTAINING |
2014 |
- Krylova Svetlana Gennad'Evna
- Amosova Evdokija Naumovna
- Zueva Elena Petrovna
- Razina Tat'Jana Georgievna
- Rybalkina Ol'Ga Jur'Evna
- Lopatina Ksenija Aleksandrovna
- Sysoljatin Sergej Viktorovich
- Kalashnikov Aleksandr Ivanovich
- Malykhin Valerij Viktorovich
- Dygaj Aleksandr Mikhajlovich
- Zhdanov Vadim Vadimovich
|
RU2558148C1 |
| 4-(3,4-DIBROMOTHIOPHENECARBONYL)-10-ISONICOTINYL-2,6,8,12-TETRAACETYL-2,4,6,8,10,12-HEXAAZATETRA-CYCLO[5,5,0,0,0]DODECANE AS AN ANALGESIC AND A METHOD OF ITS OBTAINING |
2022 |
- Baibakova Olga Vladimirovna
- Eremina Valeriia Valerevna
- Kulagina Daria Aleksandrovna
- Alekseeva Natalia Alekseevna
- Sysoliatin Sergei Viktorovich
|
RU2799639C1 |
| 4-(3,4-DIBROMOTHIOPHENECARBONIL)-2,6,8,12-TETRAACETIL-2,4,6,8,10,12-HEXAAZATETRACYCLO[5,5,0,0,0]DODECANE DERIVATIVES WITH SALICYLIC ACIDS AS ANALGESICS AND METHOD FOR THEIR PRODUCTION |
2022 |
- Baibakova Olga Vladimirovna
- Eremina Valeriia Valerevna
- Kulagina Daria Aleksandrovna
- Alekseeva Natalia Alekseevna
- Sysoliatin Sergei Viktorovich
|
RU2802003C1 |
| ONE-POT METHOD OF PRODUCING 4,10-DI(2-ETHOXYACETYL)-2,6,8,12-TETRAACETYL-2,4,6,8,10,12-HEXAAZATETRACYCLO[5,5,0,0,0]DODECANE |
2023 |
- Eremina Valeriia Valerevna
- Kulagina Daria Aleksandrovna
- Alekseeva Natalia Alekseevna
- Sysoliatin Sergei Viktorovich
|
RU2834298C1 |
